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Target
POsterior Segregation
Ligand
BDBM39354
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
10785±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM39354
Synonyms:
2,2,4-trimethyl-6-oxidanylidene-3H-pyran-5-carbonitrile | 2,2,4-trimethyl-6-oxo-3H-pyran-5-carbonitrile | 6-keto-2,2,4-trimethyl-3H-pyran-5-carbonitrile | MLS000079232 | SMR000037070 | cid_572006
Type:
Small organic molecule
Emp. Form.:
C9H11NO2
Mol. Mass.:
165.1891
SMILES:
CC1=C(C#N)C(=O)OC(C)(C)C1 |c:1|
Structure:
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