Reaction Details Report a problem with these data
Target
Calmodulin-1
Ligand
BDBM59171
Substrate
n/a
Meas. Tech.
Fluorescence spectroscopy
Kd
7e+1± 5e+1 nM
Citation
 Trevitt, CR; Craven, CJ; Milanesi, L; Syson, K; Mattinen, ML; Perkins, J; Annila, A; Hunter, CA; Waltho, JP Enhanced ligand affinity for receptors in which components of the binding site are independently mobile. Chem Biol 12:89-97 (2005) [PubMed]  Article 
Target
Name:
Calmodulin-1
Synonyms:
CALM | CALM1 | CALM1_HUMAN | CALM2 | CAM | CAM1 | CAM2 | CAMB | Calmodulin-2
Type:
Protein
Mol. Mass.:
16813.73
Organism:
Human
Description:
P0DP23
Residue:
149
Sequence:
MADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK
  
Inhibitor
Name:
BDBM59171
Synonyms:
BN1
Type:
Small organic molecule
Emp. Form.:
C26H20N2O4S2
Mol. Mass.:
488.578
SMILES:
O=S(=O)(Nc1ccc(NS(=O)(=O)c2cccc3ccccc23)cc1)c1cccc2ccccc12
Structure:
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