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Target
Trans-activator protein BZLF1
Ligand
BDBM64841
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
>67047±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64841
Synonyms:
5-[1-(4-chlorophenyl)-1,2,3,4-tetrazol-5-yl]-2-pyridin-2-yl-4-thiophen-2-yl-pyrimidine | 5-[1-(4-chlorophenyl)-1H-tetraazol-5-yl]-2-(2-pyridinyl)-4-(2-thienyl)pyrimidine | 5-[1-(4-chlorophenyl)-5-tetrazolyl]-2-(2-pyridinyl)-4-thiophen-2-ylpyrimidine | 5-[1-(4-chlorophenyl)tetrazol-5-yl]-2-(2-pyridyl)-4-(2-thienyl)pyrimidine | 5-[1-(4-chlorophenyl)tetrazol-5-yl]-2-pyridin-2-yl-4-thiophen-2-ylpyrimidine | MLS000550216 | SMR000114284 | cid_3504805
Type:
Small organic molecule
Emp. Form.:
C20H12ClN7S
Mol. Mass.:
417.874
SMILES:
Clc1ccc(cc1)-n1nnnc1-c1cnc(nc1-c1cccs1)-c1ccccn1
Structure:
Search PDB for entries with ligand similarity: