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Target
Trans-activator protein BZLF1
Ligand
BDBM64851
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
3033±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64851
Synonyms:
2-(cyclohexylcarbamoyl)-7-oxabicyclo[2.2.1]heptane-3-carboxylic acid | 2-[(cyclohexylamino)-oxomethyl]-7-oxabicyclo[2.2.1]heptane-3-carboxylic acid | 3-[(cyclohexylamino)carbonyl]-7-oxabicyclo[2.2.1]heptane-2-carboxylic acid | MLS000704826 | SMR000231207 | cid_3327313
Type:
Small organic molecule
Emp. Form.:
C14H21NO4
Mol. Mass.:
267.3208
SMILES:
[H]C12CCC([H])(O1)C(C2C(O)=O)C(=O)NC1CCCCC1 |TLB:12:7:6:3.2,THB:9:8:6:3.2|
Structure:
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