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Target
Trans-activator protein BZLF1
Ligand
BDBM64862
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5)
IC50
47562±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of PP1: fluorescence-based biochemical high throughput dose response assay to identify inhibitors of Protein Phosphatase 5 (PP5) PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM64862
Synonyms:
5-chloranyl-7-[(4-methylpiperazin-1-yl)-pyridin-2-yl-methyl]quinolin-8-ol | 5-chloro-7-[(4-methyl-1-piperazinyl)-(2-pyridinyl)methyl]-8-quinolinol | 5-chloro-7-[(4-methylpiperazin-1-yl)-pyridin-2-ylmethyl]quinolin-8-ol | 5-chloro-7-[(4-methylpiperazino)-(2-pyridyl)methyl]quinolin-8-ol | MLS000774453 | SMR000371742 | cid_3515733
Type:
Small organic molecule
Emp. Form.:
C20H21ClN4O
Mol. Mass.:
368.86
SMILES:
CN1CCN(CC1)C(c1ccccn1)c1cc(Cl)c2cccnc2c1O
Structure:
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