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Target
Bcl-2-like protein 11
Ligand
BDBM66482
Substrate
n/a
Meas. Tech.
Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis
EC50
>350000±n/a nM
Citation
 PubChem, PC Luminescence Cell-Based Dose Retest to Identify Inhibitors of A1 Apoptosis PubChem Bioassay (2010)[AID] 
Target
Name:
Bcl-2-like protein 11
Synonyms:
B2L11_HUMAN | BCL2-like 11 isoform 1 | BCL2L11 | BIM
Type:
PROTEIN
Mol. Mass.:
22175.26
Organism:
Homo sapiens (Human)
Description:
EBI_101325
Residue:
198
Sequence:
MAKQPSDVSSECDREGRQLQPAERPPQLRPGAPTSLQTEPQGNPEGNHGGEGDSCPHGSPQGPLAPPASPGPFATRSPLFIFMRRSSLLSRSSSGYFSFDTDRSPAPMSCDKSTQTPSPPCQAFNHYLSAMASMRQAEPADMRPEIWIAQELRRIGDEFNAYYARRVFLNNYQAAEDHPRMVILRLLRYIVRLVWRMH
  
Inhibitor
Name:
BDBM66482
Synonyms:
(E)-3-(4-bromophenyl)-1-[4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)phenyl]-2-propen-1-one | (E)-3-(4-bromophenyl)-1-[4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)phenyl]prop-2-en-1-one | MLS000391412 | SMR000260448 | cid_6014681
Type:
Small organic molecule
Emp. Form.:
C19H17BrN2OS
Mol. Mass.:
401.32
SMILES:
Brc1ccc(C=CC(=O)c2ccc(cc2)N=C2NCCCS2)cc1 |w:15.15,6.6|
Structure:
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