Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67420
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
15785±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67420
Synonyms:
1-(4-benzo[cd]indol-2-ylpiperazin-1-yl)ethanone | 1-(4-benzo[cd]indol-2-ylpiperazino)ethanone | 1-[4-(2-benzo[cd]indolyl)-1-piperazinyl]ethanone | MLS000057573 | SMR000060800 | cid_2328568
Type:
Small organic molecule
Emp. Form.:
C17H17N3O
Mol. Mass.:
279.3364
SMILES:
CC(=O)N1CCN(CC1)C1=Nc2cccc3cccc1c23 |t:10|
Structure:
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