Reaction Details Report a problem with these data
Target
Protein Rev
Ligand
BDBM67433
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction
IC50
>25171±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of gld-1: Fluorescence polarization-based biochemical high throughput dose response assay for inhibitors of the HIV Rev protein-RRE RNA interaction PubChem Bioassay (2010)[AID] 
Target
Name:
Protein Rev
Synonyms:
Human immunodeficiency virus type 1 REV | REV_HV1H2 | rev
Type:
PROTEIN
Mol. Mass.:
13078.11
Organism:
Human immunodeficiency virus 1
Description:
ChEMBL_79479
Residue:
116
Sequence:
MAGRSGDSDEELIRTVRLIKLLYQSNPPPNPEGTRQARRNRRRRWRERQRQIHSISERILGTYLGRSAEPVPLQLPPLERLTLDCNEDCGTSGTQGVGSPQILVESPTVLESGTKE
  
Inhibitor
Name:
BDBM67433
Synonyms:
MLS001004132 | N-(6-methoxy-3-pyridinyl)-2-phenylacetamide | N-(6-methoxy-3-pyridyl)-2-phenyl-acetamide | N-(6-methoxypyridin-3-yl)-2-phenyl-ethanamide | N-(6-methoxypyridin-3-yl)-2-phenylacetamide | SMR000377800 | cid_16196270
Type:
Small organic molecule
Emp. Form.:
C14H14N2O2
Mol. Mass.:
242.2732
SMILES:
COc1ccc(NC(=O)Cc2ccccc2)cn1
Structure:
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