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Target
Sentrin-specific protease 8
Ligand
BDBM51101
Substrate
n/a
Meas. Tech.
Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay
IC50
>100000±n/a nM
Citation
 PubChem, PC Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 8 (SENP8) using a Luminescent assay PubChem Bioassay (2010)[AID] 
Target
Name:
Sentrin-specific protease 8
Synonyms:
DEN1 | NEDP1 | PRSC2 | SENP8 | SENP8_HUMAN | SUMO/sentrin specific peptidase family member 8
Type:
Enzyme Catalytic Domain
Mol. Mass.:
24104.52
Organism:
Homo sapiens (Human)
Description:
gi_262118306
Residue:
212
Sequence:
MDPVVLSYMDSLLRQSDVSLLDPPSWLNDHIIGFAFEYFANSQFHDCSDHVSFISPEVTQFIKCTSNPAEIAMFLEPLDLPNKRVVFLAINDNSNQAAGGTHWSLLVYLQDKNSFFHYDSHSRSNSVHAKQVAEKLEAFLGRKGDKLAFVEEKAPAQQNSYDCGMYVICNTEALCQNFFRQQTESLLQLLTPAYITKKRGEWKDLITTLAKK
  
Inhibitor
Name:
BDBM51101
Synonyms:
(benzalamino)-benzo[cd]indol-2-yl-amine | MLS000392783 | N-(benzylideneamino)benzo[cd]indol-2-amine | N-[(phenylmethylene)amino]-2-benzo[cd]indolamine | N-[(phenylmethylidene)amino]benzo[cd]indol-2-amine | SMR000261715 | [(E)-benzalamino]-benzo[cd]indol-2-yl-amine | cid_2315076
Type:
Small organic molecule
Emp. Form.:
C18H13N3
Mol. Mass.:
271.3159
SMILES:
N(N=Cc1ccccc1)C1=Nc2cccc3cccc1c23 |w:1.0,t:10|
Structure:
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