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Target
Ubiquitin-conjugating enzyme E2 N
Ligand
BDBM43800
Substrate
n/a
Meas. Tech.
Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay
IC50
>20000±0 nM
Citation
 PubChem, PC Dose Response confirmation of uHTS for the identification of UBC13 Polyubiquitin Inhibitors via a TR-FRET Assay PubChem Bioassay (2011)[AID] 
Target
Name:
Ubiquitin-conjugating enzyme E2 N
Synonyms:
BLU | UBE2N | UBE2N_HUMAN | ubiquitin-conjugating enzyme E2 N
Type:
PROTEIN
Mol. Mass.:
17137.61
Organism:
Homo sapiens (Human)
Description:
EBI_101440
Residue:
152
Sequence:
MAGLPRRIIKETQRLLAEPVPGIKAEPDESNARYFHVVIAGPQDSPFEGGTFKLELFLPEEYPMAAPKVRFMTKIYHPNVDKLGRICLDILKDKWSPALQIRTVLLSIQALLSAPNPDDPLANDVAEQWKTNEAQAIETARAWTRLYAMNNI
  
Inhibitor
Name:
BDBM43800
Synonyms:
MLS-0096316.0001 | N'-[2-(4-methoxyphenoxy)-1-oxoethyl]-2-pyridinecarbohydrazide | N'-[2-(4-methoxyphenoxy)acetyl]picolinohydrazide | N'-[2-(4-methoxyphenoxy)acetyl]pyridine-2-carbohydrazide | N'-[2-(4-methoxyphenoxy)ethanoyl]pyridine-2-carbohydrazide | cid_774167
Type:
Small organic molecule
Emp. Form.:
C15H15N3O4
Mol. Mass.:
301.2973
SMILES:
COc1ccc(OCC(=O)NNC(=O)c2ccccn2)cc1
Structure:
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