Reaction Details Report a problem with these data
Target
X-box-binding protein 1
Ligand
BDBM49288
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
1030±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM49288
Synonyms:
(5-chloro-2-pyridyl)-[4-(2-thienyl)thiazol-2-yl]amine | 5-chloro-N-[4-(2-thienyl)-1,3-thiazol-2-yl]-2-pyridinamine | MLS000064746 | N-(5-chloranylpyridin-2-yl)-4-thiophen-2-yl-1,3-thiazol-2-amine | N-(5-chloro-2-pyridinyl)-4-thiophen-2-yl-2-thiazolamine | N-(5-chloropyridin-2-yl)-4-thiophen-2-yl-1,3-thiazol-2-amine | SMR000077573 | cid_2214576
Type:
Small organic molecule
Emp. Form.:
C12H8ClN3S2
Mol. Mass.:
293.795
SMILES:
Clc1ccc(Nc2nc(cs2)-c2cccs2)nc1
Structure:
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