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Target
X-box-binding protein 1
Ligand
BDBM67836
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
10000±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM67836
Synonyms:
3-(phenylcarbonyl)-2-(trifluoromethyl)benzo[f][1]benzofuran-4,9-dione | 3-benzoyl-2-(trifluoromethyl)benzo[f][1]benzofuran-4,9-dione | 3-benzoyl-2-(trifluoromethyl)benzo[f]benzofuran-4,9-dione | 3-benzoyl-2-(trifluoromethyl)benzo[f]benzofuran-4,9-quinone | 3-benzoyl-2-(trifluoromethyl)naphtho[2,3-b]furan-4,9-dione | MLS000533785 | SMR000141223 | cid_1207959
Type:
Small organic molecule
Emp. Form.:
C20H9F3O4
Mol. Mass.:
370.2783
SMILES:
FC(F)(F)c1oc2c(c1C(=O)c1ccccc1)C(=O)c1ccccc1C2=O
Structure:
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