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Target
cAMP-dependent protein kinase type II-beta regulatory subunit
Ligand
BDBM81295
Substrate
n/a
Meas. Tech.
Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex
EC50
68984±n/a nM
Citation
 PubChem, PC Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R2B (PKA-R2B) complex PubChem Bioassay (2011)[AID] 
Target
Name:
cAMP-dependent protein kinase type II-beta regulatory subunit
Synonyms:
KAP3_HUMAN | PRKAR2B
Type:
PROTEIN
Mol. Mass.:
46282.41
Organism:
Homo sapiens (Human)
Description:
EBI_11972
Residue:
418
Sequence:
MSIEIPAGLTELLQGFTVEVLRHQPADLLEFALQHFTRLQQENERKGTARFGHEGRTWGDLGAAAGGGTPSKGVNFAEEPMQSDSEDGEEEEAAPADAGAFNAPVINRFTRRASVCAEAYNPDEEEDDAESRIIHPKTDDQRNRLQEACKDILLFKNLDPEQMSQVLDAMFEKLVKDGEHVIDQGDDGDNFYVIDRGTFDIYVKCDGVGRCVGNYDNRGSFGELALMYNTPRAATITATSPGALWGLDRVTFRRIIVKNNAKKRKMYESFIESLPFLKSLEFSERLKVVDVIGTKVYNDGEQIIAQGDSADSFFIVESGEVKITMKRKGKSEVEENGAVEIARCSRGQYFGELALVTNKPRAASAHAIGTVKCLAMDVQAFERLLGPCMEIMKRNIATYEEQLVALFGTNMDIVEPTA
  
Inhibitor
Name:
BDBM81295
Synonyms:
4-{(E)-[4-(dimethylamino)-1-naphthyl]diazenyl}benzenesulfonate | MLS000719909 | SMR000304438 | cid_23679857 | sodium;4-[[4-(dimethylamino)-1-naphthalenyl]azo]benzenesulfonate | sodium;4-[[4-(dimethylamino)-1-naphthyl]azo]besylate | sodium;4-[[4-(dimethylamino)naphthalen-1-yl]diazenyl]benzenesulfonate
Type:
Small organic molecule
Emp. Form.:
C18H16N3O3S
Mol. Mass.:
354.403
SMILES:
CN(C)c1ccc(\N=N\c2ccc(cc2)S([O-])(=O)=O)c2ccccc12
Structure:
Search PDB for entries with ligand similarity: