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Target
5-hydroxytryptamine 1D receptor
Ligand
BDBM81780
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_1752
Citation
 Rinaldi-Carmona, M; Congy, C; Santucci, V; Simiand, J; Gautret, B; Neliat, G; Labeeuw, B; Le Fur, G; Soubrie, P; Breliere, JC Biochemical and pharmacological properties of SR 46349B, a new potent and selective 5-hydroxytryptamine2 receptor antagonist. J Pharmacol Exp Ther 262:759-68 (1992) [PubMed] 
Target
Name:
5-hydroxytryptamine 1D receptor
Synonyms:
5-hydroxytryptamine 1D receptor (5HT1D) | HTR1D
Type:
Protein
Mol. Mass.:
12731.52
Organism:
Bos taurus (Bovine)
Description:
Q8MI13
Residue:
119
Sequence:
SNRSLNATATQGAWDPGTLQALKIALVVLLSIITLATVLSNAFVLTTIFLTRKLHTPANCLIGSLAMTDLLVSILVMPISIAYTTTHTWSFGQLLCDIWLSSDITCCTASILHLCVIAL
  
Inhibitor
Name:
BDBM81780
Synonyms:
CAS_6438382 | NSC_6438382 | SR 46349B
Type:
Small organic molecule
Emp. Form.:
C19H21FN2O2
Mol. Mass.:
328.3806
SMILES:
CN(C)CCON=C(C=Cc1ccc(O)cc1)c1ccccc1F |w:6.5,8.7|
Structure:
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