Reaction Details
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5-hydroxytryptamine 1D receptor
Ligand
BDBM50056401
Substrate
n/a
Ki
2511.88±n/a nM
Comments
PDSP_1689
Citation
Buchheit, KH; Gamse, R; Pfannkuche, HJ SDZ 205-557, a selective, surmountable antagonist for 5-HT4 receptors in the isolated guinea pig ileum. Naunyn Schmiedebergs Arch Pharmacol 345:387-93 (1992) [PubMed] Article More Info.:
Target
Name:
5-hydroxytryptamine 1D receptor
Synonyms:
5-hydroxytryptamine 1D receptor (5HT1D) | HTR1D
Type:
Protein
Mol. Mass.:
12731.52
Organism:
Bos taurus (Bovine)
Description:
Q8MI13
Residue:
119
Sequence:
SNRSLNATATQGAWDPGTLQALKIALVVLLSIITLATVLSNAFVLTTIFLTRKLHTPANCLIGSLAMTDLLVSILVMPISIAYTTTHTWSFGQLLCDIWLSSDITCCTASILHLCVIAL
Inhibitor
Name:
BDBM50056401
Synonyms:
2-diethylaminoethyl [2-methoxy-4-amino-5-chloro]benzoate | 4-Amino-5-chloro-2-methoxy-benzoic acid 2-diethylamino-ethyl ester | CHEMBL287045 | SDZ 205557 | SDZ-205557
Type:
Small organic molecule
Emp. Form.:
C14H21ClN2O3
Mol. Mass.:
300.781
SMILES:
CCN(CC)CCOC(=O)c1cc(Cl)c(N)cc1OC
Structure:
