Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM81946
Substrate
n/a
Ki
8.8±n/a nM
Comments
PDSP_1121
Citation
 Andersen, PH The dopamine inhibitor GBR 12909: selectivity and molecular mechanism of action. Eur J Pharmacol 166:493-504 (1989) [PubMed]  Article 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM81946
Synonyms:
CAS_96850-13-4 | LU 19,005 | LU 19-005
Type:
Small organic molecule
Emp. Form.:
C16H15Cl2N
Mol. Mass.:
292.203
SMILES:
CN[C@H]1C[C@@H](c2ccccc12)c1ccc(Cl)c(Cl)c1 |r|
Structure:
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