Reaction Details Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM81987
Substrate
n/a
Ki
3.29±n/a nM
Comments
PDSP_3140
Citation
 Shank, RP; Vaught, JL; Pelley, KA; Setler, PE; McComsey, DF; Maryanoff, BE McN-5652: a highly potent inhibitor of serotonin uptake. J Pharmacol Exp Ther 247:1032-8 (1988) [PubMed] 
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM81987
Synonyms:
CHEMBL116048 | McN-5652-15
Type:
Small organic molecule
Emp. Form.:
C19H21NS
Mol. Mass.:
295.442
SMILES:
CSc1ccc(cc1)C1CN2CCCC2c2ccccc12
Structure:
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