Reaction Details Report a problem with these data
Target
Neuropeptide Y receptor type 1
Ligand
BDBM82276
Substrate
n/a
Ki
0.16±n/a nM
Comments
PDSP_1030
Citation
 Gerald, C; Walker, MW; Vaysse, PJ; He, C; Branchek, TA; Weinshank, RL Expression cloning and pharmacological characterization of a human hippocampal neuropeptide Y/peptide YY Y2 receptor subtype. J Biol Chem 270:26758-61 (1995) [PubMed]  Article 
Target
Name:
Neuropeptide Y receptor type 1
Synonyms:
NPY-Y1 | NPY1-R | NPY1R | NPY1R_HUMAN | NPYR | NPYY1 | neuropeptide Y receptor Y1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44399.07
Organism:
Homo sapiens (Human)
Description:
NPY-Y1 NPY1R HUMAN::P25929
Residue:
384
Sequence:
MNSTLFSQVENHSVHSNFSEKNAQLLAFENDDCHLPLAMIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAIMCLPFTFVYTLMDHWVFGEAMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYVGIAVIWVLAVASSLPFLIYQVMTDEPFQNVTLDAYKDKYVCFDQFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKMRDNKYRSSETKRINIMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKINNNDDNEKI
  
Inhibitor
Name:
BDBM82276
Synonyms:
L31,P34-NPY,human | NPY Leu31, Pro34, human, rat | NPY [Leu31, Pro34], human | NPY, LP, porcine | NPY,[Leu31,Pro34] | NPY,[leu31,Pro34], porcine
Type:
Small organic molecule
Emp. Form.:
C188H282N54O56S
Mol. Mass.:
4226.644
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: