Reaction Details Report a problem with these data
Target
Nicotinic acetylcholine receptor
Ligand
BDBM50026461
Substrate
n/a
Ki
1200±n/a nM
Comments
PDSP_299
Citation
 Houghtling, RA; Dávila-García, MI; Kellar, KJ Characterization of (+/-)(-)[3H]epibatidine binding to nicotinic cholinergic receptors in rat and human brain. Mol Pharmacol 48:280-7 (1995) [PubMed] 
Target
Name:
Nicotinic acetylcholine receptor
Synonyms:
Nicotinic acetylcholine receptor | n-AChR
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2478.99
Organism:
RAT
Description:
n-AChR 0 RAT::Q62594
Residue:
23
Sequence:
MTMALLGTLLLLALFGRSQGKNE
  
Inhibitor
Name:
BDBM50026461
Synonyms:
(+-)-anabasine | 3-(piperidin-2-yl)pyridine | Anabasine, (+/-) | CHEMBL280963 | anabasine
Type:
Small organic molecule
Emp. Form.:
C10H14N2
Mol. Mass.:
162.2316
SMILES:
C1CCC(NC1)c1cccnc1
Structure:
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