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Target
Transmembrane and immunoglobulin domain-containing 3
Ligand
BDBM50194153
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_2566
Citation
 van Galen, PJ; van Bergen, AH; Gallo-Rodriguez, C; Melman, N; Olah, ME; IJzerman, AP; Stiles, GL; Jacobson, KA A binding site model and structure-activity relationships for the rat A3 adenosine receptor. Mol Pharmacol 45:1101-11 (1994) [PubMed] 
Target
Name:
Transmembrane and immunoglobulin domain-containing 3
Synonyms:
ADENOSINE A3 | ADORA3 | Adora3 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
25707.75
Organism:
RAT
Description:
Q4V8H0
Residue:
232
Sequence:
MEPLLLLSLALFSDAMVMDEKVKSGVELDTASAICNYDAHYKDHTKYWCRGYFRDSCNIIAFTPNSSNRVALKDTGDQLIITVSCLVKEDTGWYWCGIQRDFARDDMDFTKLIVTDNREDRANGLSPGTSGNRTRSCKTSKAVQKAEGSRMSILIVCVLISGLGIIFLISHMSRGRRSQRNRGVTGKSINRNPQASQAPSMVSIPLTVLPKVPRQNGQQKALQWTGNATKTG
  
Inhibitor
Name:
BDBM50194153
Synonyms:
5'-CDP | CDP | CHEMBL425252 | Cytidine | Cytidine 5'-diphosphoric acid | Cytidine 5'-pyrophosphate | Cytidine, 5'-(trihydrogen pyrophosphate) | cytidine 5'-(trihydrogen diphosphate)
Type:
Small organic molecule
Emp. Form.:
C9H15N3O11P2
Mol. Mass.:
403.1764
SMILES:
Nc1ccn([C@@H]2O[C@H](COP(O)(=O)OP(O)(O)=O)[C@@H](O)[C@H]2O)c(=O)n1
Structure:
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