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Target
Dual specificity protein kinase CLK2
Ligand
BDBM50239782
Substrate
n/a
Meas. Tech.
ChEMBL_1667062 (CHEMBL4016858)
IC50
19±n/a nM
Citation
ElHady, AK; Abdel-Halim, M; Abadi, AH; Engel, M Development of Selective Clk1 and -4 Inhibitors for Cellular Depletion of Cancer-Relevant Proteins. J Med Chem 60:5377-5391 (2017) [PubMed] Article
More Info.:
Target
Name:
Dual specificity protein kinase CLK2
Synonyms:
CDC-like kinase 2 | CLK2_MOUSE | Clk2
Type:
PROTEIN
Mol. Mass.:
60021.57
Organism:
Mus musculus
Description:
ChEMBL_1502246
Residue:
499
Sequence:
MPHPRRYHSSERGSRGSYHEHYQSRKHKRRRSRSWSSSSDRTRRRRREDSYHVRSRSSYDDHSSDRRLYDRRYCGSYRRNDYSRDRGEAYYDTDFRQSYEYHRENSSYRSQRSSRRKHRRRRRRSRTFSRSSSHSSRRAKSVEDDAEGHLIYHVGDWLQERYEIVSTLGEGTFGRVVQCVDHRRGGTQVALKIIKNVEKYKEAARLEINVLEKINEKDPDNKNLCVQMFDWFDYHGHMCISFELLGLSTFDFLKDNNYLPYPIHQVRHMAFQLCQAVKFLHDNKLTHTDLKPENILFVNSDYELTYNLEKKRDERSVKSTAVRVVDFGSATFDHEHHSTIVSTRHYRAPEVILELGWSQPCDVWSIGCIIFEYYVGFTLFQTHDNREHLAMMERILGPVPSRMIRKTRKQKYFYRGRLDWDENTSAGRYVRENCKPLRRYLTSEAEDHHQLFDLIENMLEYEPAKRLTLGEALQHPFFACLRTEPPNTKLWDSSRDISR