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Target
D(2) dopamine receptor
Ligand
BDBM50013062
Substrate
n/a
Meas. Tech.
ChEBML_58550
IC50
98±n/a nM
Citation
 Neumeyer, JL; Gao, YG; Kula, NS; Baldessarini, RJ Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist. J Med Chem 33:3122-4 (1991) [PubMed]  Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
50931.60
Organism:
Rattus norvegicus (rat)
Description:
P61169
Residue:
444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFMKILHC
  
Inhibitor
Name:
BDBM50013062
Synonyms:
11-fluoro-7-propyl-(6aR)-6a,7,8,9-tetrahydro-6H-benzo[de][1,3]dioxolo[5',4':5,6]benzo[g]quinoline | CHEMBL106886
Type:
Small organic molecule
Emp. Form.:
C20H20FNO2
Mol. Mass.:
325.3767
SMILES:
CCCN1CCc2cc(F)cc-3c2[C@H]1Cc1ccc2OCOc2c-31
Structure:
Search PDB for entries with ligand similarity: