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Target
D(2) dopamine receptor
Ligand
BDBM50019879
Substrate
n/a
Meas. Tech.
ChEBML_62569
Ki
2150±n/a nM
Citation
 Harrold, MW; Chang, YA; Wallace, RA; Farooqui, T; Wallace, LJ; Uretsky, N; Miller, DD Charged analogues of chlorpromazine as dopamine antagonists. J Med Chem 30:1631-5 (1987) [PubMed]  Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D2 | DOPAMINE D2 Long | DOPAMINE D2 Short | DRD2_RAT | Dopamine D2 receptor | Dopamine2-like | Drd2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
50931.60
Organism:
Rattus norvegicus (rat)
Description:
P61169
Residue:
444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKADRPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFMKILHC
  
Inhibitor
Name:
BDBM50019879
Synonyms:
CHEMBL279905 | [3-(2-Chloro-phenothiazin-10-yl)-propyl]-trimethyl-ammonium; iodide
Type:
Small organic molecule
Emp. Form.:
C18H22ClN2S
Mol. Mass.:
333.898
SMILES:
C[N+](C)(C)CCCN1c2ccccc2Sc2ccc(Cl)cc12
Structure:
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