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Target
Adenosine receptor A1
Ligand
BDBM50022728
Substrate
n/a
Meas. Tech.
ChEBML_29612
Ki
20000±n/a nM
Citation
 Peet, NP; Dickerson, GA; Abdallah, AH; Daly, JW; Ukena, D Benzo[1,2-c:5,4-c']dipyrazoles: non-xanthine adenosine antagonists. J Med Chem 31:2034-9 (1988) [PubMed]  Article 
Target
Name:
Adenosine receptor A1
Synonyms:
AA1R_RAT | ADENOSINE A1 | ADENOSINE A1 high | ADENOSINE A1 low | Adenosine A1 receptor (A1) | Adenosine receptor | Adenosine receptors A1 | Adora1
Type:
Protein
Mol. Mass.:
36704.13
Organism:
Rattus norvegicus (rat)
Description:
n/a
Residue:
326
Sequence:
MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVTQRRAAVAIAGCWILSLVVGLTPMFGWNNLSVVEQDWRANGSVGEPVIKCEFEKVISMEYMVYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALILFLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFLKIWNDHFRCQPKPPIDEDLPEEKAED
  
Inhibitor
Name:
BDBM50022728
Synonyms:
1,7-Diethyl-3,5,8-trimethyl-1,7-dihydro-benzo[1,2-c;5,4-c']dipyrazole | CHEMBL64784
Type:
Small organic molecule
Emp. Form.:
C15H20N4
Mol. Mass.:
256.3461
SMILES:
CCn1nc(C)c2cc3c(C)nn(CC)c3c(C)c12
Structure:
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