Reaction Details Report a problem with these data
Target
Solute carrier organic anion transporter family member 1A1
Ligand
BDBM50375594
Substrate
n/a
Meas. Tech.
ChEMBL_837108 (CHEMBL2076360)
Ki
32000±n/a nM
Citation
More Info.:
Target
Name:
Solute carrier organic anion transporter family member 1A1
Synonyms:
OATP-1 | Oatp1 | Oatp1a1 | Organic anion-transporting polypeptide 1 | SO1A1_RAT | Slc21a1 | Slco1a1 | Sodium-independent organic anion transporter 1 | Solute carrier family 21 member 1
Type:
PROTEIN
Mol. Mass.:
74188.94
Organism:
Rattus norvegicus
Description:
ChEMBL_838286
Residue:
670
Sequence:
MEETEKKIATQEGRLFSKMKVFLLSLTCACLTKSLSGVYMNSMLTQIERQFDISTSVAGLINGSFEIGNLFFIVFVSYFGTKLHRPVVIGIGCVIMGLGCLLMSLPHFFMGRYEYETTISPTGNLSSNSFLCMENRTQTLKPTQDPAECVKEMKSLMWICVMVGNIIRGIGETPIVPLGISYIEDFAKSENSPLYIGILEMGKVAGPIFGLLLGSYCAQIYVDIGSVNTDDLTITPSDTRWVGAWWIGFLVCAGVNILTSIPFFFLPKALPKKGQQENVAVTKDGKVEKYGGQAREENLGITKDFLTFMKRLFCNPIYMLFILTSVLQVNGFINKFTFLPKYLEQQYGKSTAEAIFLIGVYSLPPICLGYLIGGFIMKKFKITVKKAAYLAFCLSVFEYLLFLCHFMLTCDNAAVAGLTTSYKGVQHQLHVESKVLADCNTRCSCSTNTWDPVCGDNGVAYMSACLAGCKKFVGTGTNMVFQDCSCIQSLGNSSAVLGLCKKGPECANRLQYFLILTIIISFIYSLTAIPGYMVFLRCVKSEEKSLGVGLHTFCIRVFAGIPAPVYFGALIDRTCLHWGTLKCGQRGACRMYDINSFRHIYLGLPIALRGSSYLPAFFILILMRKFQFPGDIDSSATDHTEMMLGEKESEHTDVHGSPQVENDGELKTKL