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Target
D(3) dopamine receptor
Ligand
BDBM50032643
Substrate
n/a
Meas. Tech.
ChEMBL_62295 (CHEMBL675217)
Ki
1.9±n/a nM
Citation
 Glase, SA; Corbin, AE; Pugsley, TA; Heffner, TG; Wise, LD Synthesis and dopaminergic activity of pyridine analogs of 5-hydroxy-2-(di-n-propylamino)tetralin. J Med Chem 38:3132-7 (1995) [PubMed]  Article 
Target
Name:
D(3) dopamine receptor
Synonyms:
DOPAMINE D3 | DRD3 | DRD3_HUMAN | Dopamine D3 receptor | Dopamine D3 receptor (D3) | Dopamine D3 receptor (D3R) | Dopamine receptor | Dopamine receptor (D3) | Dopamine receptor D3
Type:
n/a
Mol. Mass.:
44243.43
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
400
Sequence:
MASLSQLSSHLNYTCGAENSTGASQARPHAYYALSYCALILAIVFGNGLVCMAVLKERALQTTTNYLVVSLAVADLLVATLVMPWVVYLEVTGGVWNFSRICCDVFVTLDVMMCTASILNLCAISIDRYTAVVMPVHYQHGTGQSSCRRVALMITAVWVLAFAVSCPLLFGFNTTGDPTVCSISNPDFVIYSSVVSFYLPFGVTVLVYARIYVVLKQRRRKRILTRQNSQCNSVRPGFPQQTLSPDPAHLELKRYYSICQDTALGGPGFQERGGELKREEKTRNSLSPTIAPKLSLEVRKLSNGRLSTSLKLGPLQPRGVPLREKKATQMVAIVLGAFIVCWLPFFLTHVLNTHCQTCHVSPELYSATTWLGYVNSALNPVIYTTFNIEFRKAFLKILSC
  
Inhibitor
Name:
BDBM50032643
Synonyms:
CHEMBL105512 | N*6*,N*6*-Dipropyl-4,5,6,7-tetrahydro-benzothiazole-2,6-diamine
Type:
Small organic molecule
Emp. Form.:
C13H23N3S
Mol. Mass.:
253.407
SMILES:
CCCN(CCC)C1CCc2nc(N)sc2C1
Structure:
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