Reaction Details Report a problem with these data
Target
Ecdysone receptor/Ultraspiracle protein
Ligand
BDBM50226672
Substrate
n/a
Meas. Tech.
ChEMBL_927052 (CHEMBL3073223)
IC50
389±n/a nM
Citation
Tohidi-Esfahani, D; Lawrence, MC; Graham, LD; Hannan, GN; Simpson, AM; Hill, RJ Isoforms of the heteropteran Nezara viridula ecdysone receptor: protein characterisation, RH5992 insecticide binding and homology modelling. Pest Manag Sci 67:1457-67 (2011) [PubMed] Article
More Info.:
Target
Name:
Ecdysone receptor/Ultraspiracle protein
Synonyms:
Ecdysone receptor
Type:
n/a
Mol. Mass.:
n/a
Description:
ASSAY_ID of ChEMBL is 927052
Components:
This complex has 2 components.
Component 1
Name:
Ecdysone receptor
Synonyms:
EcR | Ecdysteroid receptor
Type:
PROTEIN
Mol. Mass.:
45167.98
Organism:
Spodoptera frugiperda
Description:
ChEMBL_106732
Residue:
403
Sequence:
MSIESRLDSLVRGKSEVKAFTGGCPSALVDTGACDTLADMRRRWYNNGGFQTLRMLEESSSEVTSSSTLGLPPAMVMSPESLASPEYGGLELWGYEDGLTTYSMAQSLGSCTMEQQQQPQQQQPQQTQPLPSMPLPMPPTTPKSENESMSSGREELSPASSVNGCSTDGEARRQKKGPAPRQQEELCLVCGDRASGYHYNALTCEGCKGFFRRSVTKNAVYICKFGHACEMDMYMRRKCQECRLKKCLAVGMRPECVVPENQCAMKRKEKKAQREKDKLPVSTTTVDDHMPPIMQCDPPPPEAARILGCLQHEVVPRFLNEKLMEQNRLKNVPPLTANQKSLIARLVWYQEGYEQPSEEDLKRVTQTWQSDEDEEESDMPFRQITEMTILTVQLIVEFAKGLP
Component 2
Name:
Ultraspiracle protein
Synonyms:
USP | Ultraspiracle protein
Type:
PROTEIN
Mol. Mass.:
31264.93
Organism:
Spodoptera frugiperda
Description:
ChEMBL_106732
Residue:
276
Sequence:
MMEPSRDSGLNLESGFMSPMSPPEMKPDTAMLDGLRDDSTPPPAFKNYPPNHPLSGSKHLCSICGDRASGKHYGVYSCEGCKGFFKRTVRKDLTYACREERNCIIDKRQRNRCQYCRYQKCLACGMKREAVQEERQRAARGTEDAHPSSSVQVQELSIERLLEMESLVADPTEEYQFLRVGPDSNVPPKFRAPVSSLCQIGNKQIAALVVWARDIPHFSSLELEDQMLLIKGSWNELLLFAIAWRSMEYLTEEREVVDSFGNRTTSPPQLMCLMPG