Reaction Details Report a problem with these data
Target
Casein kinase 1, delta tv1
Ligand
BDBM50488820
Substrate
n/a
Meas. Tech.
ChEMBL_932131 (CHEMBL3072203)
IC50
600±n/a nM
Citation
  TBA Med Chem Res 22:3247-3258 (2013)    Article 
Target
Name:
Casein kinase 1, delta tv1
Synonyms:
CSNK1D
Type:
PROTEIN
Mol. Mass.:
47258.61
Organism:
Sus scrofa
Description:
ChEMBL_106594
Residue:
415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRAADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPVSGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
  
Inhibitor
Name:
BDBM50488820
Synonyms:
CHEMBL2295952
Type:
Small organic molecule
Emp. Form.:
C22H26N8O
Mol. Mass.:
418.4948
SMILES:
CCC[C@@H](O)Nc1nc(Nc2ccc(cc2)-c2cncnc2)c2ncn(C(C)C)c2n1 |r|
Structure:
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