Reaction Details Report a problem with these data
Target
Casein kinase 1, delta tv1
Ligand
BDBM50488817
Substrate
n/a
Meas. Tech.
ChEMBL_932131 (CHEMBL3072203)
IC50
410±n/a nM
Citation
  TBA Med Chem Res 22:3247-3258 (2013)    Article 
Target
Name:
Casein kinase 1, delta tv1
Synonyms:
CSNK1D
Type:
PROTEIN
Mol. Mass.:
47258.61
Organism:
Sus scrofa
Description:
ChEMBL_106594
Residue:
415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRAADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPVSGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
  
Inhibitor
Name:
BDBM50488817
Synonyms:
CHEMBL2295945
Type:
Small organic molecule
Emp. Form.:
C23H28N8O
Mol. Mass.:
432.5214
SMILES:
CC(C)C[C@@H](O)Nc1nc(Nc2cccc(c2)-c2cncnc2)c2ncn(C(C)C)c2n1 |r|
Structure:
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