Reaction Details
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Casein kinase 1, delta tv1
Ligand
BDBM50488802
Substrate
n/a
Meas. Tech.
ChEMBL_932131 (CHEMBL3072203)
IC50
410±n/a nM
Citation
TBA Med Chem Res 22:3247-3258 (2013) Article More Info.:
Target
Name:
Casein kinase 1, delta tv1
Synonyms:
CSNK1D
Type:
PROTEIN
Mol. Mass.:
47258.61
Organism:
Sus scrofa
Description:
ChEMBL_106594
Residue:
415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRAADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPVSGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
Inhibitor
Name:
BDBM50488802
Synonyms:
CHEMBL2295951
Type:
Small organic molecule
Emp. Form.:
C18H16ClN7
Mol. Mass.:
365.82
SMILES:
CC(C)n1cnc2c(Nc3ccc(cc3)-c3cncnc3)nc(Cl)nc12
Structure:
