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Target
5-hydroxytryptamine receptor 4
Ligand
BDBM50454556
Substrate
n/a
Meas. Tech.
ChEMBL_3347 (CHEMBL619047)
Ki
1.2±n/a nM
Citation
 Soulier, JL; Yang, D; Brémont, B; Croci, T; Guzzi, U; Langlois, M Arylcarbamate derivatives of 1-piperidineethanol as potent ligands for 5-HT4 receptors. J Med Chem 40:1755-61 (1997) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 4
Synonyms:
5-HT-4 | 5-HT4 | 5-HT4L | 5-HT4S | 5-hydroxytryptamine receptor 4 | 5HT4R_RAT | Htr4 | Serotonin (5-HT) receptor | Serotonin 4 (5-HT4) receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
46117.31
Organism:
RAT
Description:
5-HT4 HTR4 RAT::Q62758
Residue:
406
Sequence:
MDRLDANVSSNEGFGSVEKVVLLTFFAMVILMAILGNLLVMVAVCRDRQLRKIKTNYFIVSLAFADLLVSVLVNAFGAIELVQDIWFYGEMFCLVRTSLDVLLTTASIFHLCCISLDRYYAICCQPLVYRNKMTPLRIALMLGGCWVIPMFISFLPIMQGWNNIGIVDVIEKRKFNHNSNSTFCVFMVNKPYAITCSVVAFYIPFLLMVLAYYRIYVTAKEHAQQIQMLQRAGATSESRPQTADQHSTHRMRTETKAAKTLCVIMGCFCFCWAPFFVTNIVDPFIDYTVPEKVWTAFLWLGYINSGLNPFLYAFLNKSFRRAFLIILCCDDERYKRPPILGQTVPCSTTTINGSTHVLRDTVECGGQWESRCHLTATSPLVAAQPVIRRPQDNDLEDSCSLKRSQS
  
Inhibitor
Name:
BDBM50454556
Synonyms:
CHEMBL2115017
Type:
Small organic molecule
Emp. Form.:
C18H28N2O3
Mol. Mass.:
320.4265
SMILES:
CCOc1ccccc1NC(=O)OCCN1C[C@H](C)C[C@@H](C)C1
Structure:
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