Target
Chromobox protein homolog 7
Ligand
BDBM50515933
Substrate
n/a
Meas. Tech.
ChEMBL_1862780 (CHEMBL4363636)
Kd
2800±n/a nM
Citation
 Yang, LLiu, YFan, MZhu, GJin, HLiang, JLiu, ZHuang, ZZhang, L Identification and characterization of benzo[d]oxazol-2(3H)-one derivatives as the first potent and selective small-molecule inhibitors of chromodomain protein CDYL. Eur J Med Chem 182:0 (2019) [PubMed]  Article 
Target
Name:
Chromobox protein homolog 7
Synonyms:
Chromobox protein homolog 7 | CBX7_HUMAN | CBX7 | Chromobox protein homolog 7 (CBX7)
Type:
Protein
Mol. Mass.:
28351.76
Organism:
Human
Description:
n/a
Residue:
251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEKEERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKAGAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAPDVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAAEGFFRDRSGKF
  
Inhibitor
Name:
BDBM50515933
Synonyms:
CHEMBL4469115
Type:
Small organic molecule
Emp. Form.:
TBD
Mol. Mass.:
TBD
SMILES:
TBD
Structure:
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