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Target
Casein kinase 1, delta tv1
Ligand
BDBM50364141
Substrate
n/a
Meas. Tech.
ChEMBL_1985499 (CHEMBL4618905)
IC50
7.7±n/a nM
Citation
 Cescon, E; Bolcato, G; Federico, S; Bissaro, M; Valentini, A; Ferlin, MG; Spalluto, G; Sturlese, M; Moro, S Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 ? Inhibitors. ACS Med Chem Lett 11:1168-1174 (2020) [PubMed]  Article 
Target
Name:
Casein kinase 1, delta tv1
Synonyms:
CSNK1D
Type:
PROTEIN
Mol. Mass.:
47258.61
Organism:
Sus scrofa
Description:
ChEMBL_106594
Residue:
415
Sequence:
MELRVGNRYRLGRKIGSGSFGDIYLGTDIAAGEEVAIKLECVKTKHPQLHIESKIYKMMQGGVGIPTIRWCGAEGDYNVMVMELLGPSLEDLFNFCSRKFSLKTVLLLADQMISRIEYIHSKNFIHRDVKPDNFLMGLGKKGNLVYIIDFGLAKKYRDARTHQHIPYRENKNLTGTARYASINTHLGIEQSRRDDLESLGYVLMYFNLGSLPWQGLKAATKRQKYERISEKKMSTPIEVLCKGYPSEFATYLNFCRSLRFDDKPDYSYLRQLFRNLFHRQGFSYDYVFDWNMLKFGASRAADDAERERRDREERLRHSRNPATRGLPSTASGRLRGTQEAAPPTPLTPTSHTANTSPRPVSGMERERKVSMRLHRGAPVNISSSDLTGRQDTSRMSTSQIAGRVAASGLQSAVHR
  
Inhibitor
Name:
BDBM50364141
Synonyms:
CHEMBL1951415
Type:
Small organic molecule
Emp. Form.:
C19H20FN5
Mol. Mass.:
337.394
SMILES:
Nc1nccc(n1)-c1c(ncn1C1CCCCC1)-c1ccc(F)cc1
Structure:
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