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Target
Fusion glycoprotein F0
Ligand
BDBM50542662
Substrate
n/a
Meas. Tech.
ChEMBL_1987321 (CHEMBL4620868)
EC50
0.501187±n/a nM
Citation
Vendeville, S; Tahri, A; Hu, L; Demin, S; Cooymans, L; Vos, A; Kwanten, L; Van den Berg, J; Battles, MB; McLellan, JS; Koul, A; Raboisson, P; Roymans, D; Jonckers, THM Discovery of 3-({5-Chloro-1-[3-(methylsulfonyl)propyl]-1 J Med Chem 63:8046-8058 (2020) [PubMed] Article
More Info.:
Target
Name:
Fusion glycoprotein F0
Synonyms:
F | Fusion glycoprotein F0
Type:
PROTEIN
Mol. Mass.:
63485.30
Organism:
Human respiratory syncytial virus
Description:
ChEMBL_106144
Residue:
574
Sequence:
MELPILKANAITTILAAVTFCFASSQNITEEFYQSTCSAVSKGYLSALRTGWYTSVITIELSNIKENKCNGTDAKVKLMKQELDKYKNAVTELQLLMQSTPAANNRARRELPRFMNYTLNNTKKTNVTLSKKRKRRFLGFLLGVGSAIASGIAVSKVLHLEGEVNKIKSALLSTNKAVVSLSNGVSVLTSKVLDLKNYIDKQLLPIVNKQSCRISNIETVIEFQQKNNRLLEITREFSVNAGVTTPVSTYMLTNSELLSLINDMPITNDQKKLMSNNVQIVRQQSYSIMSIIKEEVLAYVVQLPLYGVIDTPCWKLHTSPLCTTNTKEGSNICLTRTDRGWYCDNAGSVSFFPQAETCKVQSNRVFCDTMNSLTLPSEVNLCNVDIFNPKYDCKIMTSKTDVSSSVITSLGAIVSCYGKTKCTASNKNRGIIKTFSNGCDYVSNKGVDTVSVGNTLYYVNKQEGKSLYVKGEPIINFYDPLVFPSDEFDASISQVNEKINQSLAFIRKSDELLHNVNAGKSTTNIMITTIIIVIIVILLSLIAVGLLLYCKARSTPVTLSKDQLSGINNIAFSN