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Target
Death-associated protein kinase 2
Ligand
BDBM50554817
Substrate
n/a
Meas. Tech.
ChEMBL_2050824 (CHEMBL4705523)
IC50
22±n/a nM
Citation
Chen, J; Zhou, Y; Dong, X; Liu, L; Bai, L; McEachern, D; Przybranowski, S; Yang, CY; Stuckey, J; Li, X; Wen, B; Zhao, T; Sun, S; Sun, D; Jiao, L; Jing, Y; Guo, M; Yang, D; Wang, S Discovery of CJ-2360 as a Potent and Orally Active Inhibitor of Anaplastic Lymphoma Kinase Capable of Achieving Complete Tumor Regression. J Med Chem 63:13994-14016 (2020) [PubMed] Article
More Info.:
Target
Name:
Death-associated protein kinase 2
Synonyms:
DAP kinase 2 | DAP-kinase-related protein 1 | DAPK2 | DAPK2_HUMAN | DRP-1
Type:
PROTEIN
Mol. Mass.:
42900.09
Organism:
Homo sapiens (Human)
Description:
ChEMBL_774557
Residue:
370
Sequence:
MFQASMRSPNMEPFKQQKVEDFYDIGEELGSGQFAIVKKCREKSTGLEYAAKFIKKRQSRASRRGVSREEIEREVSILRQVLHHNVITLHDVYENRTDVVLILELVSGGELFDFLAQKESLSEEEATSFIKQILDGVNYLHTKKIAHFDLKPENIMLLDKNIPIPHIKLIDFGLAHEIEDGVEFKNIFGTPEFVAPEIVNYEPLGLEADMWSIGVITYILLSGASPFLGDTKQETLANITAVSYDFDEEFFSQTSELAKDFIRKLLVKETRKRLTIQEALRHPWITPVDNQQAMVRRESVVNLENFRKQYVRRRWKLSFSIVSLCNHLTRSLMKKVHLRPDEDLRNCESDTEEDIARRKALHPRRRSSTS