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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50560829
Substrate
n/a
Meas. Tech.
ChEMBL_2073593 (CHEMBL4729127)
EC50
12±n/a nM
Citation
 Nakamura, S; Sayama, M; Uwamizu, A; Jung, S; Ikubo, M; Otani, Y; Kano, K; Omi, J; Inoue, A; Aoki, J; Ohwada, T Non-naturally Occurring Regio Isomer of Lysophosphatidylserine Exhibits Potent Agonistic Activity toward G Protein-Coupled Receptors. J Med Chem 63:9990-10029 (2020) [PubMed]  Article 
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
G protein-coupled receptor 34 | GPR34_MOUSE | Gpr34 | Probable G-protein coupled receptor 34
Type:
PROTEIN
Mol. Mass.:
43201.40
Organism:
Mus musculus
Description:
ChEMBL_102842
Residue:
375
Sequence:
MTTTSVDSWLCSSHGMHFITNYSDQASQNFSGVPNVTSCPMDEKLLSTVLTTFYSVIFLVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAVADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRRAITTKQSIYVCCIVWTVALAGFLTMIILTLKKGGHNSTMCFHYRDRHNAKGEAIFNFVLVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIIHKTNEIMLVFSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQSEASRSESTSEFKPGHSLHDLSVTVKMPQYSTKGN
  
Inhibitor
Name:
BDBM50560829
Synonyms:
CHEMBL4784581
Type:
Small organic molecule
Emp. Form.:
C27H48NO9P
Mol. Mass.:
561.6451
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](COCC#C)OP(O)(=O)OC[C@H](N)C(O)=O |r|
Structure:
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