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Target
Putative P2Y purinoceptor 10
Ligand
BDBM50560843
Substrate
n/a
Meas. Tech.
ChEMBL_2073596 (CHEMBL4729130)
EC50
26±n/a nM
Citation
 Nakamura, S; Sayama, M; Uwamizu, A; Jung, S; Ikubo, M; Otani, Y; Kano, K; Omi, J; Inoue, A; Aoki, J; Ohwada, T Non-naturally Occurring Regio Isomer of Lysophosphatidylserine Exhibits Potent Agonistic Activity toward G Protein-Coupled Receptors. J Med Chem 63:9990-10029 (2020) [PubMed]  Article 
Target
Name:
Putative P2Y purinoceptor 10
Synonyms:
P2Y10 | P2Y10_MOUSE | P2ry10 | Putative P2Y purinoceptor 10
Type:
PROTEIN
Mol. Mass.:
37264.07
Organism:
Mus musculus
Description:
ChEMBL_109764
Residue:
328
Sequence:
MGSNSTSSAESNCNATYLPFQYSLYATTYIFIFIPGLLANSAALWVLCRFISKKNKAIIFMINLSVADLAHILSLPLRIYYYINRHWPFQRALCLLCFYLKYLNMYASIFFLTCISLQRCLFLLKPFRARNWKRRYDVGISAVIWIVVGTACLPFPILRNAGLANSTDSCFADLGYKQMDAVVLVTMVVIAELAGFVIPVITIACCTWKTTVSLKHPPIAFQGISERKKALRMVFMCAAVFVICFTPYHINFIFYTMVKESIITSCPTVKSTLYFHPFSLCLASLCCLLDPILYYFMASEFRDQLSRHGSSVTRSRLMSRESGSSMVN
  
Inhibitor
Name:
BDBM50560843
Synonyms:
CHEMBL4759297
Type:
Small organic molecule
Emp. Form.:
C28H46NO10P
Mol. Mass.:
587.6393
SMILES:
CCCCCCCCCCCOc1ccccc1CCC(=O)O[C@@H]1COCC[C@H]1OP(O)(=O)OC[C@H](N)C(O)=O |r|
Structure:
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