Reaction Details Report a problem with these data
Target
Proteasome subunit beta type-5
Ligand
BDBM50587104
Substrate
n/a
Meas. Tech.
ChEMBL_2170916 (CHEMBL5056050)
IC50
>100000±n/a nM
Citation
Zhang, H; Hsu, HC; Kahne, SC; Hara, R; Zhan, W; Jiang, X; Burns-Huang, K; Ouellette, T; Imaeda, T; Okamoto, R; Kawasaki, M; Michino, M; Wong, TT; Toita, A; Yukawa, T; Moraca, F; Vendome, J; Saha, P; Sato, K; Aso, K; Ginn, J; Meinke, PT; Foley, M; Nathan, CF; Darwin, KH; Li, H; Lin, G Macrocyclic Peptides that Selectively Inhibit the J Med Chem 64:6262-6272 (2021) [PubMed] Article
More Info.:
Target
Name:
Proteasome subunit beta type-5
Synonyms:
20S proteasome chymotrypsin-like | 26S proteosome | LMPX | MB1 | PSB5_HUMAN | PSMB5 | Proteasome Macropain subunit MB1 | Proteasome subunit beta type-1/beta type-5 | X
Type:
Protein
Mol. Mass.:
28480.96
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
263
Sequence:
MALASVLERPLPVNQRGFFGLGGRADLLDLGPGSLSDGLSLAAPGWGVPEEPGIEMLHGTTTLAFKFRHGVIVAADSRATAGAYIASQTVKKVIEINPYLLGTMAGGAADCSFWERLLARQCRIYELRNKERISVAAASKLLANMVYQYKGMGLSMGTMICGWDKRGPGLYYVDSEGNRISGATFSVGSGSVYAYGVMDRGYSYDLEVEQAYDLARRAIYQATYRDAYSGGAVNLYHVREDGWIRVSSDNVADLHEKYSGSTP