Reaction Details Report a problem with these data
Target
G protein-activated inward rectifier potassium channel 2
Ligand
BDBM50593373
Substrate
n/a
Meas. Tech.
ChEMBL_2208118 (CHEMBL5121067)
EC50
>30000±n/a nM
Citation
Sharma, S; Lesiak, L; Aretz, CD; Du, Y; Kumar, S; Gautam, N; Alnouti, Y; Dhuria, NV; Chhonker, YS; Weaver, CD; Hopkins, CR Discovery, synthesis and biological characterization of a series of RSC Med Chem 12:1366-1373 (2021) [PubMed]
More Info.:
Target
Name:
G protein-activated inward rectifier potassium channel 2
Synonyms:
BIR1 | GIRK-2 | GIRK2 | Inward rectifier K(+) channel Kir3.2 | KATP-2 | KATP2 | KCNJ6 | KCNJ6_HUMAN | KCNJ7 | Potassium channel, inwardly rectifying subfamily J member 6
Type:
PROTEIN
Mol. Mass.:
48440.73
Organism:
Homo sapiens (Human)
Description:
ChEMBL_107630
Residue:
423
Sequence:
MAKLTESMTNVLEGDSMDQDVESPVAIHQPKLPKQARDDLPRHISRDRTKRKIQRYVRKDGKCNVHHGNVRETYRYLTDIFTTLVDLKWRFNLLIFVMVYTVTWLFFGMIWWLIAYIRGDMDHIEDPSWTPCVTNLNGFVSAFLFSIETETTIGYGYRVITDKCPEGIILLLIQSVLGSIVNAFMVGCMFVKISQPKKRAETLVFSTHAVISMRDGKLCLMFRVGDLRNSHIVEASIRAKLIKSKQTSEGEFIPLNQTDINVGYYTGDDRLFLVSPLIISHEINQQSPFWEISKAQLPKEELEIVVILEGMVEATGMTCQARSSYITSEILWGYRFTPVLTLEDGFYEVDYNSFHETYETSTPSLSAKELAELASRAELPLSWSVSSKLNQHAELETEEEEKNLEEQTERNGDVANLENESKV