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Target
Probable G-protein coupled receptor 174
Ligand
BDBM50601665
Substrate
n/a
Meas. Tech.
ChEMBL_2237843 (CHEMBL5151739)
EC50
13±n/a nM
Citation
 Sayama, M; Uwamizu, A; Ikubo, M; Chen, L; Yan, G; Otani, Y; Inoue, A; Aoki, J; Ohwada, T Switching Lysophosphatidylserine G Protein-Coupled Receptor Agonists to Antagonists by Acylation of the Hydrophilic Serine Amine. J Med Chem 64:10059-10101 (2021) [PubMed] 
Target
Name:
Probable G-protein coupled receptor 174
Synonyms:
GP174_MOUSE | Gm376 | Gpr174
Type:
PROTEIN
Mol. Mass.:
38774.65
Organism:
Mus musculus
Description:
ChEMBL_116800
Residue:
335
Sequence:
MTDNFTCNKTDGDNTDFRYFIYAVTYTVILVPGLIGNILALWVFYGYMKETKRAVVFMINLAIADLLQILSLPLRIFYYLNHDWPFGPGLCMFCFYLKYVNMYASIYFLVCISVRRFWFLMYPFRFNDCKQKYDLYISIIGWLIICLACLLFPLLRTNDDTPGNRTKCFVDLPIRNVNLAQSVAMITIGEVVGFVTPLMIVLYCTWKTALSLQNKYPISQHLGEKKKALKMILTCAGVFLVCFVPYHFSFPLDFLVKSNEIKSCFARRVILIFHSVALCLASLNSCLDPVIYYFTTNEFRRRLSRQDLPDNIQLHTKSYKIASNHATSTVAAELC
  
Inhibitor
Name:
BDBM50601665
Synonyms:
CHEMBL5202832
Type:
Small organic molecule
Emp. Form.:
C33H49N2O10P
Mol. Mass.:
664.7233
SMILES:
CCCCCCCCCCCOc1cccc(CCC(=O)NC[C@@H](O)COP(O)(=O)OC[C@H](NC(=O)c2ccccc2)C(O)=O)c1 |r|
Structure:
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