Reaction Details Report a problem with these data
Target
Sigma intracellular receptor 2
Ligand
BDBM50009307
Substrate
n/a
Meas. Tech.
ChEMBL_2243690 (CHEMBL5157900)
Ki
58±n/a nM
Citation
Bechthold, E; Schreiber, JA; Ritter, N; Grey, L; Schepmann, D; Daniliuc, C; González-Cano, R; Nieto, FR; Seebohm, G; Wünsch, B Synthesis of tropane-based ? Eur J Med Chem 230:0 (2022) [PubMed]
More Info.:
Target
Name:
Sigma intracellular receptor 2
Synonyms:
S2r | SGMR2_RAT | Sigma intracellular receptor 2 | Sigma-2 receptor | Sigma2 receptor | Tmem97 | Transmembrane protein 97
Type:
Protein
Mol. Mass.:
20953.88
Organism:
Rattus norvegicus (Rat)
Description:
Q5U3Y7
Residue:
176
Sequence:
MGAVTARRCVEWLLGLYFVSHIPITMFIDLQALLPPELYPQEFSNLLRWYSKEFKDPLMQEPPVWFKSFLFCELVFQLPFFPIAAYAFFKGSCRWIRIPAIIYAVHTITTLIPILYTILFEDFSKAIAFKGQRPENFRERLTLVGVYAPYLIIPLILLLFMLRNPYYKFEEKRKKK