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Target
B1 bradykinin receptor
Ligand
BDBM50214792
Substrate
n/a
Meas. Tech.
ChEMBL_39983 (CHEMBL653557)
EC50
85±n/a nM
Citation
 Tancredi, M; Galoppini, C; Meini, S; Quartara, L; Maggi, CA; Rovero, P Synthesis and biological activity of new bradykinin pseudopeptide B1 receptor agonists containing alkylic spacers Bioorg Med Chem Lett 7:2661-2664 (1997)    Article 
Target
Name:
B1 bradykinin receptor
Synonyms:
B1 BRADYKININ | B1R | B1bkr | BK-1 receptor | BKRB1_RAT | Bdkrb1 | Bkr | Bradykinin B1 receptor | KB1 | Kinin B1 receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38389.97
Organism:
RAT
Description:
B1 BRADYKININ BDKRB1 RAT::P97583
Residue:
337
Sequence:
MASEVLLELQPSNRSLQAPANITSCESALEDWDLLYRVLPGFVITICFFGLLGNLLVLSFFLLPWRQWWWQQRQRQQRLTIAEIYLANLAASDLVFVLGLPFWAENIGNRFNWPFGTDLCRVVSGVIKANLFVSIFLVVAISQDRYRLLVYPMTSWGYRRRRQAQATCLLIWVAGGLLSIPTFLLRSVKVVPDLNVSACILLFPHEAWHFARMVELNVLGFLLPVTAIIFFNYHILASLRGQKEASRTRCGGPKGSKTTGLILTLVASFLVCWCPYHFFAFLDFLVQVRVIQDCSWKEITDLGLQLANFFAFVNSCLNPLIYVFAGRLLKTRVLGTL
  
Inhibitor
Name:
BDBM50214792
Synonyms:
CHEMBL264100 | des-Arg10-Kallidin
Type:
Small organic molecule
Emp. Form.:
C50H73N13O11
Mol. Mass.:
1032.1951
SMILES:
NCCCC[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(O)=O
Structure:
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