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Target
Macrophage scavenger receptor types I and II
Ligand
BDBM50292391
Substrate
n/a
Meas. Tech.
ChEMBL_550891 (CHEMBL997334)
IC50
71000±n/a nM
Citation
 Freyer, AJ; Patil, AD; Killmer, L; Zuber, G; Myers, C; Johnson, RK Rigidone, a sesquiterpene o-quinone from the gorgonian Pseudopterogorgia rigida. J Nat Prod 60:309-11 (1997) [PubMed]  Article 
Target
Name:
Macrophage scavenger receptor types I and II
Synonyms:
CD_antigen=CD204 | MSR1 | MSRE_HUMAN | Macrophage acetylated LDL receptor I and II | Macrophage scavenger receptor types I and II | SCARA1 | Scavenger receptor class A member 1
Type:
PROTEIN
Mol. Mass.:
49756.01
Organism:
Homo sapiens (Human)
Description:
ChEMBL_101341
Residue:
451
Sequence:
MEQWDHFHNQQEDTDSCSESVKFDARSMTALLPPNPKNSPSLQEKLKSFKAALIALYLLVFAVLIPLIGIVAAQLLKWETKNCSVSSTNANDITQSLTGKGNDSEEEMRFQEVFMEHMSNMEKRIQHILDMEANLMDTEHFQNFSMTTDQRFNDILLQLSTLFSSVQGHGNAIDEISKSLISLNTTLLDLQLNIENLNGKIQENTFKQQEEISKLEERVYNVSAEIMAMKEEQVHLEQEIKGEVKVLNNITNDLRLKDWEHSQTLRNITLIQGPPGPPGEKGDRGPTGESGPRGFPGPIGPPGLKGDRGAIGFPGSRGLPGYAGRPGNSGPKGQKGEKGSGNTLTPFTKVRLVGGSGPHEGRVEILHSGQWGTICDDRWEVRVGQVVCRSLGYPGVQAVHKAAHFGQGTGPIWLNEVFCFGRESSIEECKIRQWGTRACSHSEDAGVTCTL
  
Inhibitor
Name:
BDBM50292391
Synonyms:
(S)-1-methyl-4-(6-methylhept-5-en-2-yl)phenazine-2,3-diol | CHEMBL463299
Type:
Small organic molecule
Emp. Form.:
C21H24N2O2
Mol. Mass.:
336.4275
SMILES:
[#6]-[#6@@H](-[#6]-[#6]\[#6]=[#6](\[#6])-[#6])-c1c(-[#8])c(-[#8])c(-[#6])c2nc3ccccc3nc12 |r|
Structure:
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