Reaction Details Report a problem with these data
Target
Growth factor receptor-bound protein 7
Ligand
BDBM50334297
Substrate
n/a
Meas. Tech.
ChEMBL_699661 (CHEMBL1648304)
Kd
5760±n/a nM
Citation
Ambaye, ND; Gunzburg, MJ; Lim, RC; Price, JT; Wilce, MC; Wilce, JA Benzopyrazine derivatives: A novel class of growth factor receptor bound protein 7 antagonists. Bioorg Med Chem 19:693-701 (2011) [PubMed] Article
More Info.:
Target
Name:
Growth factor receptor-bound protein 7
Synonyms:
B47 | Epidermal growth factor receptor GRB-7 | GRB7 | GRB7 adapter protein | GRB7_HUMAN
Type:
PROTEIN
Mol. Mass.:
59700.56
Organism:
Homo sapiens (Human)
Description:
ChEMBL_699661
Residue:
532
Sequence:
MELDLSPPHLSSSPEDLCPAPGTPPGTPRPPDTPLPEEVKRSQPLLIPTTGRKLREEERRATSLPSIPNPFPELCSPPSQSPILGGPSSARGLLPRDASRPHVVKVYSEDGACRSVEVAAGATARHVCEMLVQRAHALSDETWGLVECHPHLALERGLEDHESVVEVQAAWPVGGDSRFVFRKNFAKYELFKSSPHSLFPEKMVSSCLDAHTGISHEDLIQNFLNAGSFPEIQGFLQLRGSGRKLWKRFFCFLRRSGLYYSTKGTSKDPRHLQYVADVNESNVYVVTQGRKLYGMPTDFGFCVKPNKLRNGHKGLRIFCSEDEQSRTCWLAAFRLFKYGVQLYKNYQQAQSRHLHPSCLGSPPLRSASDNTLVAMDFSGHAGRVIENPREALSVALEEAQAWRKKTNHRLSLPMPASGTSLSAAIHRTQLWFHGRISREESQRLIGQQGLVDGLFLVRESQRNPQGFVLSLCHLQKVKHYLILPSEEEGRLYFSMDDGQTRFTDLLQLVEFHQLNRGILPCLLRHCCTRVAL