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Target
PHD finger protein 13
Ligand
BDBM50341830
Substrate
n/a
Meas. Tech.
ChEMBL_743694 (CHEMBL1767463)
IC50
48000±n/a nM
Citation
 Herold, JM; Wigle, TJ; Norris, JL; Lam, R; Korboukh, VK; Gao, C; Ingerman, LA; Kireev, DB; Senisterra, G; Vedadi, M; Tripathy, A; Brown, PJ; Arrowsmith, CH; Jin, J; Janzen, WP; Frye, SV Small-molecule ligands of methyl-lysine binding proteins. J Med Chem 54:2504-11 (2011) [PubMed]  Article 
Target
Name:
PHD finger protein 13
Synonyms:
PHF13 | PHF13_HUMAN | SPOC1 | Survival time-associated PHD finger protein in ovarian cancer 1
Type:
PROTEIN
Mol. Mass.:
33585.46
Organism:
Homo sapiens (Human)
Description:
ChEMBL_743694
Residue:
300
Sequence:
MDSDSCAAAFHPEEYSPSCKRRRTVEDFNKFCTFVLAYAGYIPYPKEELPLRSSPSPANSTAGTIDSDGWDAGFSDIASSVPLPVSDRCFSHLQPTLLQRAKPSNFLLDRKKTDKLKKKKKRKRRDSDAPGKEGYRGGLLKLEAADPYVETPTSPTLQDIPQAPSDPCSGWDSDTPSSGSCATVSPDQVKEIKTEGKRTIVRQGKQVVFRDEDSTGNDEDIMVDSDDDSWDLVTCFCMKPFAGRPMIECNECHTWIHLSCAKIRKSNVPEVFVCQKCRDSKFDIRRSNRSRTGSRKLFLD
  
Inhibitor
Name:
BDBM50341830
Synonyms:
5-Bromo-N-(5-(pyrrolidin-1-yl)pentylnicotinamide | CHEMBL1767022
Type:
Small organic molecule
Emp. Form.:
C15H22BrN3O
Mol. Mass.:
340.259
SMILES:
Brc1cncc(c1)C(=O)NCCCCCN1CCCC1
Structure:
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