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Target
Cytohesin-3
Ligand
BDBM50075651
Substrate
n/a
Meas. Tech.
ChEMBL_787633 (CHEMBL1918086)
Kd
100±n/a nM
Citation
 Anraku, K; Inoue, T; Sugimoto, K; Kudo, K; Okamoto, Y; Morii, T; Mori, Y; Otsuka, M Design and synthesis of biotinylated inositol 1,3,4,5-tetrakisphosphate targeting Grp1 pleckstrin homology domain. Bioorg Med Chem 19:6833-41 (2011) [PubMed]  Article 
Target
Name:
Cytohesin-3
Synonyms:
PH, SEC7 and coiled-coil domain-containing protein 3 | SEC7 homolog C | rSec7-3 | CYH3_RAT | Cyth3 | Pscd3 | Sec7c
Type:
PROTEIN
Mol. Mass.:
46329.05
Organism:
Rat
Description:
ChEMBL_787633
Residue:
400
Sequence:
MDEGGGGEGGSVPEDLSLEEREELLDIRRRKKELIDDIERLKYEIAEVMTEIDNLTSVEESKTTQRNKQIAMGRKKFNMDPKKGIQFLIENDLLQSSPEDVAQFLYKGEGLNKTVIGDYLGERDDFNIKVLQAFVELHEFADLNLVQALRQFLWSFRLPGEAQKIDRMMEAFASRYCLCNPGVFQSTDTCYVLSFAIIMLNTSLHNHNVRDKPTAERFITMNRGINEGGDLPEELLRNLYESIKNEPFKIPEDDGNDLTHTFFNPDREGWLLKLGGGRVKTWKRRWFILTDNCLYYFEYTTDKEPRGIIPLENLSIREVEDPRKPNCFELYNPSHKGQVIKACKTEADGRVVEGNHVVYRISAPSPEEKEEWMKSIKASISRDPFYDMLATRKRRIANKK
  
Inhibitor
Name:
BDBM50075651
Synonyms:
1D-myo-inositol 1,3,4,5-tetrakis(dihydrogen phosphate) | 1D-myo-inositol 1,3,4,5-tetrakisphosphate | CHEMBL23552
Type:
Small organic molecule
Emp. Form.:
n/a
Mol. Mass.:
n/a
SMILES:
[C@H]1([C@H](C([C@H]([C@H](C1OP(=O)(O)O)O)OP(=O)(O)O)OP(=O)(O)O)OP(=O)(O)O)O
Structure:
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