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Target
Mu-type opioid receptor
Ligand
BDBM50326659
Substrate
n/a
Meas. Tech.
ChEBML_138742
Ki
0.700000±n/a nM
Citation
 Schmidhammer, H; Stangl, A; Furst, Z; Szabo, E; Borsodi, A; Patel, D; Traynor, JR Synthesis and biological evaluation of 14-alkoxymorphinans.12.1 A phenethyl analogue of the -selective opioid receptor antagonist cyprodime Bioorg Med Chem Lett 5:1923-1926 (1995)    Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50326659
Synonyms:
3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one | 3,10-dimethoxy-17-methyl-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-13-one | CHEMBL606644
Type:
Small organic molecule
Emp. Form.:
C19H25NO3
Mol. Mass.:
315.4067
SMILES:
COc1cccc2C[C@H]3N(C)CC[C@@]4(CC(=O)CC[C@@]34OC)c12 |r|
Structure:
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