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Target
Mu-type opioid receptor
Ligand
BDBM50098194
Substrate
n/a
Meas. Tech.
ChEBML_145297
Ki
30±n/a nM
Citation
 Clayson, J; Jales, A; Tyacke, RJ; Hudson, AL; Nutt, DJ; Lewis, JW; Husbands, SM Selective delta-opioid receptor ligands: potential PET ligands based on naltrindole. Bioorg Med Chem Lett 11:939-43 (2001) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50098194
Synonyms:
11-(2-fluoroethyl)-22-methyl-(2S)-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5(10),6,8,15(25),16,18-heptaene-2,16-diol | CHEMBL435898
Type:
Small organic molecule
Emp. Form.:
C25H25FN2O3
Mol. Mass.:
420.476
SMILES:
CN1CCC23[C@H]4Oc5c2c(CC1[C@]3(O)Cc1c4n(CCF)c2ccccc12)ccc5O |TLB:13:12:8.9.10:1.3.2,0:1:12:8.9.10,THB:7:8:12:1.3.2|
Structure:
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