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Target
N-acetyllactosaminide alpha-1,3-galactosyltransferase
Ligand
BDBM50367549
Substrate
n/a
Meas. Tech.
ChEBML_219109
Ki
165000±n/a nM
Citation
 Vaghefi, MM; Bernacki, RJ; Dalley, NK; Wilson, BE; Robins, RK Synthesis of glycopyranosylphosphonate analogues of certain natural nucleoside diphosphate sugars as potential inhibitors of glycosyltransferases. J Med Chem 30:1383-91 (1987) [PubMed]  Article 
Target
Name:
N-acetyllactosaminide alpha-1,3-galactosyltransferase
Synonyms:
GGTA1_MOUSE | Galactosyltransferase | Ggta-1 | Ggta1 | UDP-galactose:beta-D-galactosyl-1,4-N-acetyl-D-glucosaminide alpha-1,3-galactosyltransferase
Type:
PROTEIN
Mol. Mass.:
46474.57
Organism:
Mus musculus
Description:
ChEMBL_219109
Residue:
394
Sequence:
MITMLQDLHVNKISMSRSKSETSLPSSRSGSQEKIMNVKGKVILLMLIVSTVVVVFWEYVNRIPEVGENRWQKDWWFPSWFKNGTHSYQEDNVEGRREKGRNGDRIEEPQLWDWFNPKNRPDVLTVTPWKAPIVWEGTYDTALLEKYYATQKLTVGLTVFAVGKYIEHYLEDFLESADMYFMVGHRVIFYVMIDDTSRMPVVHLNPLHSLQVFEIRSEKRWQDISMMRMKTIGEHILAHIQHEVDFLFCMDVDQVFQDNFGVETLGQLVAQLQAWWYKASPEKFTYERRELSAAYIPFGEGDFYYHAAIFGGTPTHILNLTRECFKGILQDKKHDIEAQWHDESHLNKYFLFNKPTKILSPEYCWDYQIGLPSDIKSVKVAWQTKEYNLVRNNV
  
Inhibitor
Name:
BDBM50367549
Synonyms:
CHEMBL604428
Type:
Small organic molecule
Emp. Form.:
C15H24N2O16P2
Mol. Mass.:
550.3024
SMILES:
OC[C@H]1OC([C@H](O)[C@@H](O)[C@@H]1O)P(O)(=O)OP(O)(=O)OC[C@H]1OC([C@H](O)[C@@H]1O)n1ccc(=O)[nH]c1=O |r|
Structure:
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