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Target
3',5'-cyclic-AMP phosphodiesterase
Ligand
BDBM50020874
Substrate
n/a
Meas. Tech.
ChEMBL_155847 (CHEMBL766943)
IC50
37200±n/a nM
Citation
 Takase, Y; Saeki, T; Fujimoto, M; Saito, I Cyclic GMP phosphodiesterase inhibitors. 1. The discovery of a novel potent inhibitor, 4-((3,4-(methylenedioxy)benzyl)amino)-6,7,8-trimethoxyquinazoline. J Med Chem 36:3765-70 (1994) [PubMed]  Article 
Target
Name:
3',5'-cyclic-AMP phosphodiesterase
Synonyms:
Phosphodiesterase 4A
Type:
PROTEIN
Mol. Mass.:
13615.65
Organism:
Sus scrofa
Description:
ChEMBL_155848
Residue:
118
Sequence:
PWLVGWWDQFKRMLNRELTHLSEMSRSGNQVSEYISTTFLDKQNEVDIPSPTMKDHEKQQAPRQRPSQQPPPPGPQFQPMSQITGVKKLMHSSSLNEDSSIPRFGVKTDQEELLAQEL
  
Inhibitor
Name:
BDBM50020874
Synonyms:
(3-Chloro-phenyl)-(4-phenyl-phthalazin-1-yl)-amine | CHEMBL332898
Type:
Small organic molecule
Emp. Form.:
C20H14ClN3
Mol. Mass.:
331.798
SMILES:
Clc1cccc(Nc2nnc(-c3ccccc3)c3ccccc23)c1
Structure:
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